SCHEMBL3720526

SCHEMBL3720526

CCOC(=O)c1cc(-c2cccs2)nc(-c2ccc(C#Cc3cccnc3)cc2)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.49
KDM4E B2RXH2 7/20 0.49
HPGD P15428 5/20 0.49
GAA P10253 4/20 0.49
CASP1 P29466 1/20 0.49
MAPT P10636 6/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GRM5 P41594 1/20 0.42
GLA P06280 1/20 0.41
RECQL P46063 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 1/20 0.39
UBE2I P63279 2/20 0.39
SAE1 Q9UBE0 2/20 0.39
UBA2 Q9UBT2 2/20 0.39
CDC7 O00311 1/20 0.38
DBF4 Q9UBU7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720782 0.91 MEN1 (0.47) ALDH1A1KDM4EHPGDGAACASP1
SCHEMBL3713520 0.89 GRM5 (0.46) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL13188838 0.86 MAPT (0.40) ALDH1A1KDM4EHPGDGAAMAPT
SCHEMBL3712449 0.86 GRM5 (0.44) ALDH1A1KDM4EHPGDGAACASP1
SCHEMBL3713434 0.86 GRM5 (0.48) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL3713522 0.85 GRM5 (0.43) ALDH1A1KDM4EHPGDCASP1MAPT
SCHEMBL3710606 0.83 GRM5 (0.42) ALDH1A1KDM4EHPGDMAPTMEN1
SCHEMBL3711244 0.83 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDGAACASP1
SCHEMBL3710598 0.80 GRM5 (0.42) ALDH1A1KDM4EHPGDMAPTLMNA
SCHEMBL3709730 0.77 PLA2G2A (0.44) ALDH1A1KDM4EHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed