SCHEMBL3711249

SCHEMBL3711249

O=C(N1CCc2ccccc2CC1)C(F)(F)F.O=C(OC(=O)C(F)(F)F)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 2/20 0.52
ESR1 P03372 4/20 0.51
ESR2 Q92731 4/20 0.51
NOTUM Q6P988 1/20 0.45
MAPT P10636 2/20 0.44
TAAR1 Q96RJ0 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
ACE P12821 1/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
RIPK1 Q13546 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3711251 1.00 ABHD6 (0.52) ABHD6ESR1ESR2NOTUMMAPT
SCHEMBL5908776 0.93 ABHD6 (0.59) ABHD6ESR1ESR2NOTUMMAPT
SCHEMBL5908773 0.93 ABHD6 (0.59) ABHD6ESR1ESR2NOTUMMAPT
SCHEMBL506139 0.90 ESR1 (0.59) ABHD6ESR1ESR2NOTUMMAPT
SCHEMBL566389 0.82 ESR1 (0.68) ABHD6ESR1ESR2NOTUMMAPT
SCHEMBL30263783 0.82 ESR1 (0.68) ABHD6ESR1ESR2NOTUMMAPT
SCHEMBL373718 0.75 ESR1 (0.58) ABHD6ESR1ESR2
SCHEMBL7368230 0.75 MTNR1B (0.50) ESR1ESR2MEN1KMT2AACE
SCHEMBL506963 0.74 ESR1 (0.50) ABHD6ESR1ESR2
SCHEMBL5424954 0.73 RIPK1 (0.72) ABHD6ESR1ESR2NOTUMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096384-A2 FUSED BENZAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2010-08-26 WO disclosed