SCHEMBL3711295

SCHEMBL3711295

COCCNc1nc2c(C)c(F)ccc2cc1CCNC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 4/20 0.39
RXFP1 Q9HBX9 1/20 0.39
PIK3CD O00329 4/20 0.37
GRM1 Q13255 1/20 0.37
CSNK2A1 P68400 1/20 0.35
HSD17B10 Q99714 3/20 0.35
CASP7 P55210 3/20 0.34
LMNA P02545 2/20 0.34
TSHR P16473 2/20 0.34
CASP1 P29466 2/20 0.34
MAPK1 P28482 1/20 0.34
HCAR3 P49019 1/20 0.34
USP2 O75604 2/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3705670 0.80 PIK3CD (0.43) ALDH1A1KDM4EPIK3CDGRM1TSHR
SCHEMBL7307 0.79 ALDH1A1 (0.40) ALDH1A1KDM4EHSD17B10LMNATSHR
SCHEMBL863915 0.79 CDK5 (0.39) ALDH1A1KDM4ERXFP1CSNK2A1MAPK1
SCHEMBL3711291 0.78 ALDH1A1 (0.35) ALDH1A1KDM4ERXFP1PIK3CDCSNK2A1
SCHEMBL3714054 0.75 KDM4E (0.37) ALDH1A1KDM4ERXFP1PIK3CDHSD17B10
SCHEMBL3714056 0.75 KDM4E (0.37) ALDH1A1KDM4ERXFP1PIK3CDHSD17B10
SCHEMBL7863 0.68 PIK3CD (0.38) ALDH1A1KDM4EPIK3CDHSD17B10TSHR
SCHEMBL20562599 0.68 MTNR1A (0.56) MTNR1AMTNR1B
SCHEMBL23291226 0.67 MAPT (0.48) ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL15184778 0.66 HTR7 (0.39) ALDH1A1KDM4ERXFP1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396315-A1 FUSED PYRIDINE AND PYRAZINE DERIVATIVES AS KINASE INHIBITORS UCB Pharma, S.A. (BE) 2011-12-21 EP disclosed
WO-2010092340-A1 FUSED PYRIDINE AND PYRAZINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-08-19 WO disclosed