SCHEMBL3712909

SCHEMBL3712909

COCCNc1cc(C(=O)OC)cc(Cl)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.46
ALDH1A1 P00352 3/20 0.44
CDC7 O00311 1/20 0.43
ROCK2 O75116 1/20 0.43
PIM1 P11309 1/20 0.43
PRKACA P17612 1/20 0.43
CDK2 P24941 1/20 0.43
GSK3B P49841 1/20 0.43
CDK7 P50613 1/20 0.43
CDK9 P50750 1/20 0.43
HIPK2 Q9H2X6 1/20 0.43
IRAK4 Q9NWZ3 1/20 0.43
KDM4E B2RXH2 4/20 0.42
HPGD P15428 1/20 0.41
PTGER4 P35408 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1579303 0.84 KDM4D (0.46) ALDH1A1CDC7ROCK2PIM1PRKACA
SCHEMBL3715043 0.83 HRH4 (0.46) ALDH1A1KDM4ECA12CA1CA2
SCHEMBL569249 0.79 ALDH1A1 (0.59) ALDH1A1KDM4EHPGDCA12CA1
SCHEMBL3854836 0.78 ALDH1A1 (0.43) ALDH1A1KDM4ECA12CA1CA2
SCHEMBL3712550 0.78 HCAR3 (0.42) HCAR3ALDH1A1CDC7ROCK2PIM1
SCHEMBL3715743 0.78 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDCA12CA1
Hydrochloric Acid SCHEMBL29890892 0.77 ALDH1A1 (0.57) ALDH1A1KDM4EHPGDCA12CA1
SCHEMBL13116015 0.76 CDC7 (0.47) HCAR3ALDH1A1CDC7ROCK2PIM1
SCHEMBL4819595 0.76 CDC7 (0.47) HCAR3ALDH1A1CDC7ROCK2PIM1
SCHEMBL3711270 0.76 PIK3CA (0.61) ALDH1A1GSK3BCDK7CDK9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed