SCHEMBL3714023

SCHEMBL3714023

Cc1ccccc1-c1cccc(C(N)=O)c1NCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD38 P28907 1/20 0.50
RPS6KB1 P23443 3/20 0.46
AURKA O14965 2/20 0.46
CYP1A2 P05177 3/20 0.44
CYP2D6 P10635 3/20 0.44
TSHR P16473 3/20 0.44
CYP2C19 P33261 3/20 0.44
MYC P01106 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 1/20 0.44
ALOX15 P16050 1/20 0.44
KMT2A Q03164 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
FFAR1 O14842 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
SCN5A Q14524 1/20 0.43
SCN2A Q99250 1/20 0.43
JAK2 O60674 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3698508 0.85 MYC (0.44) CD38RPS6KB1AURKAMYCALDH1A1
SCHEMBL3704894 0.82 ALDH1A1 (0.48) CD38RPS6KB1AURKAMYCALDH1A1
SCHEMBL3708751 0.80 HTT (0.43) CD38RPS6KB1AURKATSHRMYC
SCHEMBL5482149 0.76 MYC (0.47) CD38MYCALDH1A1ALOX15KMT2A
SCHEMBL1788703 0.74 BCAT2 (0.59) TSHRMYCALDH1A1KMT2AKDM4E
SCHEMBL6131490 0.74 GSK3B (0.48) CD38RPS6KB1KMT2AKDM4ECLK4
SCHEMBL7739113 0.73 CDC7 (0.43) CD38RPS6KB1AURKACLK4CDC7
SCHEMBL5742619 0.73 MYC (0.53) TSHRMYCALDH1A1KDM4EHPGD
SCHEMBL30311518 0.73 HSD17B10 (0.63) CD38RPS6KB1AURKAALDH1A1KMT2A
SCHEMBL3135445 0.73 MYC (0.53) CYP1A2TSHRMYCCYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed