SCHEMBL3714823

SCHEMBL3714823

NN(c1ccncc1)N1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 2/20 0.48
ADRB2 P07550 1/20 0.48
NCF1 P14598 1/20 0.48
CYP2D6 P10635 3/20 0.37
CYP3A4 P08684 2/20 0.37
SLC6A4 P31645 1/20 0.36
HPGD P15428 1/20 0.35
CHRM5 P08912 1/20 0.34
CHKA P35790 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
PRKCB P05771 1/20 0.33
PRKCA P17252 1/20 0.33
PRKCH P24723 1/20 0.33
PRKCE Q02156 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28228488 0.81 SIGMAR1 (0.45)
Dalfampridine SCHEMBL28141942 0.71 ADRB2 (0.46) PLD1ADRB2NCF1CYP2D6CYP3A4
SCHEMBL4173238 0.71 ADRB2 (0.42) PLD1ADRB2NCF1CYP2D6CYP3A4
SCHEMBL894239 0.66 ADRB2 (1.00) PLD1ADRB2NCF1CYP2D6CYP3A4
SCHEMBL74335 0.66 ADRB2 (1.00) PLD1ADRB2NCF1CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL639824 0.64 ADRB2 (0.96) PLD1ADRB2NCF1CYP2D6CYP3A4
Methylpiperazine SCHEMBL28292988 0.64 CYP2D6 (0.50) PLD1ADRB2NCF1CYP2D6CYP3A4
SCHEMBL12893509 0.64 MKNK1 (0.53) HPGDTSHRCHRNB2CHRNA4
Bromide SCHEMBL9067259 0.63 ADRB2 (0.92) PLD1ADRB2NCF1CYP2D6CYP3A4
SCHEMBL22086464 0.62 CHRM5 (0.52) CYP2D6HPGDCHRM5CHKAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398795-A1 HETEROARYL SUBSTITUTED PYRIDAZINONE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-12-28 EP disclosed
WO-2010094762-A1 HETEROARYL SUBSTITUTED PYRIDAZINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-08-26 WO disclosed