SCHEMBL3715319

SCHEMBL3715319

COC(=O)Cc1cc2c(C(F)(F)F)cccc2[nH]c1=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.44
KDM4E B2RXH2 4/20 0.41
LMNA P02545 1/20 0.41
PARP1 P09874 2/20 0.41
HSD17B10 Q99714 3/20 0.40
KMT2A Q03164 1/20 0.40
NR3C1 P04150 1/20 0.39
DAO P14920 2/20 0.39
DDO Q99489 2/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
AR P10275 2/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
SRC P12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31146189 0.79 DYRK1A (0.38) EGFRKDM4ELMNAPARP1KMT2A
SCHEMBL3716515 0.76 KDM4E (0.40) KDM4ELMNAHSD17B10KMT2AALDH1A1
SCHEMBL8306652 0.75 KDM4E (0.59) KDM4EHSD17B10KMT2AALDH1A1HPGD
SCHEMBL24190146 0.74 ABL1 (0.46) KDM4EHSD17B10KMT2ANR3C1ALDH1A1
SCHEMBL30396884 0.74 ABL1 (0.46) KDM4EHSD17B10KMT2ANR3C1ALDH1A1
SCHEMBL3359175 0.73 DAO (0.64) KDM4ELMNAKMT2ADAODDO
SCHEMBL871601 0.72 POLQ (0.55) KDM4EALDH1A1
SCHEMBL30474543 0.72 POLQ (0.55) KDM4EALDH1A1
SCHEMBL31645683 0.72 P2RX7 (0.47) KDM4E
SCHEMBL31146101 0.72 EGFR (0.40) EGFRKDM4ELMNAHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393806-A1 INHIBITORS OF JUN N-TERMINAL KINASE Elan Pharmaceuticals Inc. (US) 2011-12-14 EP disclosed
WO-2010091310-A1 INHIBITORS OF JUN N-TERMINAL KINASE ELAN PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed