SCHEMBL3716745

SCHEMBL3716745

CC(C)COc1ccc(Oc2ccc3cc(CC=O)ccc3n2)cc1Br

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.35
TLR8 Q9NR97 1/20 0.35
SCN9A Q15858 8/20 0.34
ACACB O00763 1/20 0.33
SCN7A Q01118 3/20 0.32
KCNH2 Q12809 3/20 0.32
SCN5A Q14524 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN8A Q9UQD0 1/20 0.32
PDE10A Q9Y233 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
GPR55 Q9Y2T6 1/20 0.31
PDE4B Q07343 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3717217 0.89 LMNA (0.36) SCN9ASCN7AKCNH2SCN5ASCN2A
SCHEMBL3716838 0.89 ACACB (0.33) XDHTLR8SCN9AACACBSCN7A
SCHEMBL3721301 0.88 PPARG (0.35) TLR8ACACBSCN7AKCNH2SCN5A
SCHEMBL3719990 0.86 LMNA (0.37) XDHTLR8SCN9AACACBSCN7A
SCHEMBL3719435 0.86 TLR8 (0.37) XDHTLR8SCN9AACACBALDH1A1
SCHEMBL3719552 0.83 PDE3B (0.34) XDHACACBALDH1A1MAPTHDAC1
SCHEMBL3727015 0.83 PPARG (0.35) SCN9AACACBSCN7AKCNH2PDE4B
SCHEMBL3724297 0.82 ACACB (0.38) TLR8ACACBPDE10AALDH1A1MAPT
SCHEMBL3721410 0.82 MAPT (0.36) PDE10AALDH1A1MAPTTHRB
SCHEMBL3716743 0.82 PDE4B (0.49) XDHTLR8SCN9AACACBSCN7A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed