SCHEMBL3717233

SCHEMBL3717233

CC(C)(c1cccc(I)c1)S(C)(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 7/20 0.35
PDE4A P27815 3/20 0.34
PDE4B Q07343 3/20 0.34
PDE4C Q08493 3/20 0.34
PDE4D Q08499 3/20 0.34
KAT6A Q92794 1/20 0.33
LMNA P02545 1/20 0.33
PMP22 Q01453 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NR3C2 P08235 1/20 0.33
TP53BP1 Q12888 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
FAAH O00519 1/20 0.32
MGLL Q99685 1/20 0.32
HTR2C P28335 1/20 0.31
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17571915 0.78 ACHE (0.42) CYP2C9LMNA
SCHEMBL30515572 0.77 TSHR (0.48) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL25329184 0.77 CA1 (0.51) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL17560554 0.77 TSHR (0.48) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL18243516 0.75 FAAH (0.39) TP53BP1HDAC4HDAC2HDAC8FAAH
SCHEMBL12161965 0.74 NR3C2 (0.47) NR3C2HDAC4HDAC2HDAC8
SCHEMBL134474 0.74 HDAC8 (0.47) CYP2C9HDAC4HDAC2HDAC8
SCHEMBL30486770 0.73 RXRA (0.49)
SCHEMBL16094358 0.73 RXRA (0.49)
SCHEMBL26811585 0.73 ESR1 (0.34) TP53BP1HDAC4HDAC2HDAC8FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396295-A1 PHENOXY ACETIC ACID DERIVATIVES Merck Serono S.A. (CH) 2011-12-21 EP disclosed
WO-2010092043-A1 PHENOXY ACETIC ACID DERIVATIVES MERCK SERONO S.A. (CH) 2010-08-19 WO disclosed
US-5208259-A Lipoxygenase enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES (GB) 1993-05-04 US disclosed
EP-0409413-A2 Diaryl ether heterocycles IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-01-23 EP disclosed