SCHEMBL3718481

SCHEMBL3718481

COc1ccc(Oc2ccc3cc(C(C)=O)ccc3n2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.54
NNMT P40261 1/20 0.43
HPGDS O60760 6/20 0.43
HPGD P15428 2/20 0.42
PPARG P37231 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
ALDH1A1 P00352 1/20 0.41
F2 P00734 1/20 0.41
GLA P06280 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
SCN9A Q15858 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3725359 0.82 PDE4B (0.49) PDE4BHPGDSSCN9ASCN10A
SCHEMBL3720127 0.82 PDE4B (0.49) PDE4BHPGDSCYP3A4SCN9ASCN10A
SCHEMBL3717735 0.81 PDE4B (0.57) PDE4BHPGDSHPGDALDH1A1F2
SCHEMBL3717384 0.79 PDE4B (0.53) PDE4BALDH1A1SCN9ASMN1; SMN2
SCHEMBL3724294 0.79 PDE4B (0.55) PDE4BHPGDCYP1A2CYP3A4ALDH1A1
SCHEMBL3717123 0.78 ACACB (0.50)
SCHEMBL3719988 0.78 PDE4B (0.53) PDE4BHPGDALDH1A1SCN9ANPC1
SCHEMBL3717125 0.78 MTNR1A (0.64) SCN9ASMN1; SMN2MEN1KMT2ASCN10A
SCHEMBL3720702 0.78 PDE4B (0.57) PDE4BHPGDPPARGALDH1A1GLA
SCHEMBL3718630 0.78 PDE4B (0.54) PDE4BALDH1A1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed