SCHEMBL3720127

SCHEMBL3720127

CC(=O)c1ccc2nc(Oc3ccc(NC(C)C)nc3)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.49
HCAR3 P49019 1/20 0.45
HPGDS O60760 1/20 0.41
SCN9A Q15858 14/20 0.38
PDE10A Q9Y233 1/20 0.38
SCN10A Q9Y5Y9 2/20 0.37
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
FPR2 P25090 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720024 0.84 PDE4B (0.53) PDE4BHPGDSSCN9A
SCHEMBL3722765 0.83 ACACB (0.45) SCN9A
SCHEMBL3718481 0.82 PDE4B (0.54) PDE4BHPGDSSCN9ASCN10ACYP3A4
SCHEMBL3722768 0.81 MTNR1A (0.50) SCN9A
SCHEMBL3721952 0.80 SCN9A (0.37) HCAR3SCN9ASCN10A
SCHEMBL3720074 0.80 JAK2 (0.36) HCAR3SCN9A
SCHEMBL3720129 0.80 ACACB (0.37) HCAR3SCN9A
SCHEMBL3723898 0.79 PDE4B (0.50) PDE4B
SCHEMBL3725359 0.79 PDE4B (0.49) PDE4BHPGDSSCN9ASCN10A
SCHEMBL3724294 0.78 PDE4B (0.55) PDE4BSCN9ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed