SCHEMBL3720032

SCHEMBL3720032

Clc1nnc2ccc(Oc3cccc(CN4CCOCC4)c3)nn12

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 2/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
NCF1 P14598 1/20 0.43
BRD4 O60885 1/20 0.42
LMNA P02545 1/20 0.40
MET P08581 2/20 0.40
CYP3A4 P08684 2/20 0.40
HRH3 Q9Y5N1 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TRPV6 Q9H1D0 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
PDE4B Q07343 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14832703 0.81 PDE4B (0.49) ALDH1A1KDM4EHPGDHTTCYP3A4
SCHEMBL3729185 0.76 MET (0.59) ALDH1A1KDM4EHPGDHTTMET
SCHEMBL18596494 0.74 L3MBTL1 (0.67) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL16439068 0.74 L3MBTL1 (0.48) ALDH1A1KDM4EHTTLMNACYP3A4
SCHEMBL16428752 0.73 SLC2A1 (0.39) KDM4EL3MBTL1
SCHEMBL17099378 0.73 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDHTTNCF1
SCHEMBL14832474 0.73 LRRK2 (0.56) ALDH1A1KDM4EHPGDHTTBRD4
SCHEMBL14832950 0.72 LRRK2 (0.49) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL14832883 0.71 SMN1; SMN2 (0.50) ALDH1A1KDM4EHPGDHTTLMNA
SCHEMBL16439060 0.71 LRRK2 (0.69) ALDH1A1KDM4EHPGDCYP3A4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393791-A1 DERIVATIVES OF 6-(6-O-SUBSTITUTED-TRIAZOLOPYRIDAZINE-SULFANYL) BENZOTHIAZOLES AND BENZIMIDAZOLES, PREPARATION THEREOF, USE THEREOF AS DRUGS, AND USE THEREOF AS MET INHIBITORS SANOFI (FR) 2011-12-14 EP disclosed
WO-2010089507-A1 DERIVATIVES OF 6-(6-O-SUBSTITUTED-TRIAZOLOPYRIDAZINE-SULFANYL) BENZOTHIAZOLES AND BENZIMIDAZOLES, PREPARATION THEREOF, USE THEREOF AS DRUGS, AND USE THEREOF AS MET INHIBITORS SANOFI-AVENTIS (FR) 2010-08-12 WO disclosed