SCHEMBL3720175

SCHEMBL3720175

CC(Br)Oc1cccc(OC(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.41
SLC6A4 P31645 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
GPR139 Q6DWJ6 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
CETP P11597 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
CYP2C9 P11712 1/20 0.38
ACACB O00763 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14446352 0.85 PTPN5 (0.46) HDAC8GPR139ALDH1A1GAAMAPT
SCHEMBL17911612 0.84 MTNR1A (0.40) ALDH1A1GAAHTT
SCHEMBL3155575 0.81 CETP (0.43) TAS1R3TAS1R1TAS1R2GPR139ALDH1A1
SCHEMBL3147185 0.80 GPR3 (0.50) CETPCHRM2CHRM1CHRM3
SCHEMBL11748337 0.79 PPARG (0.49) ALDH1A1GAAMAPT
SCHEMBL21831249 0.79 SLC6A4 (0.45) HDAC8SLC6A4GPR139CETPCHRM2
SCHEMBL29699129 0.79 SLC6A4 (0.45) HDAC8SLC6A4GPR139CETPCHRM2
SCHEMBL8370452 0.78 GPR139 (0.43) HDAC8GPR139CETPCYP2C9
SCHEMBL4572866 0.77 MTNR1A (0.50) ALDH1A1
SCHEMBL5270292 0.77 KCNH2 (0.47) ALDH1A1GAAMAPTHPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed