SCHEMBL3720441

SCHEMBL3720441

CC(=O)c1ccc(N2CCN(c3nc(CN)cc(-c4ccc(C(F)(F)F)cc4)n3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
SCN9A Q15858 1/20 0.41
PARP1 P09874 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
CYP11B2 P19099 2/20 0.41
SLC6A7 Q99884 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CETP P11597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3725420 0.86 HSD17B10 (0.50) MAPTSMN1; SMN2PARP1PARP2HRH4
SCHEMBL3720439 0.85 KDM4E (0.53) MAPTSMN1; SMN2HPGDHTTNPC1
SCHEMBL3724664 0.82 HRH4 (0.57) MAPTSMN1; SMN2HPGDHTTHRH4
SCHEMBL3797918 0.80 HRH4 (0.44) SMN1; SMN2HPGDHRH4CYP11B2TP53
SCHEMBL3718066 0.79 HRH4 (0.43) MAPTSMN1; SMN2HPGDHRH4CYP11B2
SCHEMBL3722161 0.79 HRH4 (0.53) MAPTSMN1; SMN2HPGDHTTHRH4
SCHEMBL3720932 0.78 IDH2 (0.44) HPGDPOLBHRH4TP53
SCHEMBL3721777 0.78 HRH3 (0.42) SMN1; SMN2HPGDHRH4CYP11B2TP53
SCHEMBL3721072 0.78 CYP11B2 (0.46) MAPTSMN1; SMN2HPGDHRH4CYP11B2
SCHEMBL3724736 0.76 TRPV1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed