SCHEMBL3722006

SCHEMBL3722006

COc1ccc(Oc2cnc(CNC(=O)C3(N)CCOC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
EPHX2 P34913 7/20 0.37
MAPK10 P53779 7/20 0.36
MAPK8 P45983 3/20 0.36
PDE4B Q07343 1/20 0.36
CNR2 P34972 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722862 0.91 P2RX7 (0.43) P2RX7EPHX2MAPK10MAPK8
SCHEMBL2787523 0.88 L3MBTL1 (0.43) P2RX7EPHX2L3MBTL1KMT2A
Hydrochloric Acid SCHEMBL2788143 0.88 L3MBTL1 (0.42) P2RX7EPHX2L3MBTL1KMT2A
SCHEMBL13191711 0.86 P2RX7 (0.37) P2RX7EPHX2MAPK10MAPK8PDE4B
SCHEMBL3728281 0.86 P2RX7 (0.38) P2RX7EPHX2MAPK10MAPK8PDE4B
SCHEMBL3722075 0.85 P2RX7 (0.37) P2RX7EPHX2MAPK10MAPK8PDE4B
SCHEMBL13165651 0.84 MAPT (0.45) P2RX7EPHX2L3MBTL1KMT2A
SCHEMBL13191712 0.83 BDKRB1 (0.38) P2RX7EPHX2PDE4BCNR2
SCHEMBL3722055 0.83 P2RX7 (0.35) P2RX7EPHX2MAPK8PDE4BCNR2
SCHEMBL3725868 0.82 MEN1 (0.41) P2RX7EPHX2PDE4BCNR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed