SCHEMBL3728281

SCHEMBL3728281

COc1ccc(Oc2cnc(CNC(=O)C3(NC(=O)C(F)(F)F)CCOC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
EPHX2 P34913 9/20 0.35
CNR1 P21554 1/20 0.34
BDKRB1 P46663 1/20 0.34
PDE4B Q07343 1/20 0.34
CNR2 P34972 1/20 0.33
TP53 P04637 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK10 P53779 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
MMP1 P03956 1/20 0.33
MMP13 P45452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13191711 0.91 P2RX7 (0.37) P2RX7EPHX2PDE4BCNR2TP53
SCHEMBL3722075 0.91 P2RX7 (0.37) P2RX7EPHX2BDKRB1PDE4BCNR2
SCHEMBL13191712 0.89 BDKRB1 (0.38) P2RX7EPHX2BDKRB1PDE4BCNR2
SCHEMBL3722055 0.89 P2RX7 (0.35) P2RX7EPHX2PDE4BCNR2MAPK8
SCHEMBL3725868 0.88 MEN1 (0.41) P2RX7EPHX2BDKRB1PDE4BCNR2
SCHEMBL3721990 0.87 BDKRB1 (0.37) P2RX7EPHX2CNR1BDKRB1PDE4B
SCHEMBL3722006 0.86 P2RX7 (0.40) P2RX7EPHX2PDE4BCNR2MAPK8
SCHEMBL13165640 0.82 L3MBTL1 (0.41) P2RX7EPHX2
SCHEMBL3725821 0.81 P2RX7 (0.40) P2RX7EPHX2BDKRB1MAPK8MAPK10
SCHEMBL13165638 0.80 EPHX2 (0.40) P2RX7EPHX2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed