SCHEMBL3722356

SCHEMBL3722356

CC(=O)N(C)c1ccc(Nc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.60
L3MBTL1 Q9Y468 2/20 0.56
MAPT P10636 4/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TDP1 Q9NUW8 2/20 0.52
ALDH1A1 P00352 2/20 0.52
MAPK1 P28482 1/20 0.52
CASP7 P55210 1/20 0.52
POLB P06746 1/20 0.52
WNK1 Q9H4A3 1/20 0.49
AKR1C3 P42330 2/20 0.47
AKR1C2 P52895 2/20 0.47
ALDH3A1 P30838 2/20 0.47
AKR1B10 O60218 1/20 0.47
AKR1B1 P15121 1/20 0.47
AKR1C4 P17516 1/20 0.47
AKR1C1 Q04828 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11744600 0.83 MAPT (0.64) HCAR3MAPTNPSR1ALDH1A1MAPK1
SCHEMBL3720192 0.79 HCAR3 (0.59) HCAR3MAPTNPSR1ALDH1A1MAPK1
SCHEMBL11341363 0.79 HCAR3 (0.79) HCAR3L3MBTL1MAPTTDP1ALDH1A1
SCHEMBL3719024 0.77 HCAR3 (0.61) HCAR3MAPTNPSR1TDP1ALDH1A1
SCHEMBL109353 0.77 TDP1 (0.67) HCAR3L3MBTL1MAPTTDP1ALDH1A1
SCHEMBL2338616 0.75 HCAR3 (1.00) HCAR3L3MBTL1MAPTALDH1A1POLB
SCHEMBL3719487 0.75 HCAR3 (0.62) HCAR3MAPTNPSR1TDP1ALDH1A1
SCHEMBL11877200 0.75 ALDH1A1 (0.57) HCAR3MAPTNPSR1TDP1ALDH1A1
SCHEMBL4967065 0.75 MAPT (0.48) HCAR3L3MBTL1MAPTNPSR1TDP1
SCHEMBL1437915 0.75 HCAR3 (0.68) HCAR3L3MBTL1MAPTTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010126922-A1 BENZIMIDAZOLECARBOXAMIDES AS INHIBITORS OF FAK GLAXOSMITHKLINE LLC (US) 2010-11-04 WO disclosed
WO-2010126922-A1 BENZIMIDAZOLECARBOXAMIDES AS INHIBITORS OF FAK GLAXOSMITHKLINE LLC (US) 2010-11-04 WO disclosed