SCHEMBL3722600

SCHEMBL3722600

CCCCCc1cc(N)c2c(n1)[nH]c1ccc(-c3ccc(OCCCN(CC)CC)cc3)cc12

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AGER Q15109 4/20 0.40
PIM1 P11309 2/20 0.40
HRH3 Q9Y5N1 7/20 0.39
ATP4A P20648 3/20 0.39
ATP4B P51164 3/20 0.39
XDH P47989 1/20 0.39
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3433146 0.86 ATP4A (0.41) AGERHRH3ATP4AATP4BACHE
SCHEMBL676481 0.85 HRH2 (0.49) HRH3ACHE
SCHEMBL3423187 0.84 AGER (0.41) AGERPIM1HRH3ATP4AATP4B
SCHEMBL674976 0.82 DRD3 (0.43) AGER
SCHEMBL3725266 0.82 ALK (0.40) AGERPIM1HRH3ATP4AATP4B
SCHEMBL3426131 0.82 ATP4A (0.39) AGERPIM1HRH3ATP4AATP4B
SCHEMBL675732 0.81 KDM4E (0.43)
SCHEMBL3426129 0.80 DRD2 (0.39) PIM1HRH3ATP4AATP4BPIM2
SCHEMBL3433144 0.79 HRH3 (0.40) AGERHRH3ATP4AATP4BACHE
SCHEMBL3432969 0.77 LSS (0.42) HRH3ATP4AATP4BACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed