SCHEMBL3433146

SCHEMBL3433146

CCCCCc1ccc2c(n1)[nH]c1ccc(-c3ccc(OCCCN(CC)CC)cc3)cc12

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 1/20 0.41
ATP4B P51164 1/20 0.41
AGER Q15109 6/20 0.40
HRH3 Q9Y5N1 4/20 0.40
ACHE P22303 2/20 0.40
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3426129 0.92 DRD2 (0.39) ATP4AATP4BHRH3ACHEDRD2
SCHEMBL3432969 0.91 LSS (0.42) ATP4AATP4BHRH3ACHE
SCHEMBL3722601 0.88 HRH3 (0.41) ATP4AATP4BHRH3ACHEDRD2
SCHEMBL3423190 0.87 HRH3 (0.40) ATP4AATP4BHRH3ACHEDRD2
SCHEMBL3722600 0.86 AGER (0.40) ATP4AATP4BAGERHRH3ACHE
SCHEMBL3426135 0.84 HRH3 (0.39) ATP4AATP4BHRH3ACHEDRD2
SCHEMBL3423187 0.84 AGER (0.41) ATP4AATP4BAGERHRH3ACHE
SCHEMBL3426131 0.84 ATP4A (0.39) ATP4AATP4BAGERHRH3ACHE
SCHEMBL674726 0.84 ACHE (0.46) ATP4AATP4BAGERHRH3ACHE
SCHEMBL3724896 0.84 CCNB2 (0.44) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed