SCHEMBL3723955

SCHEMBL3723955

O=C(O)N1CCC(n2c(=O)[nH]c3ncccc32)C[C@@H]1CCCN(Cc1ccccc1)Cc1ccccc1.O=C(O)NCCCn1c(=O)[nH]c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 5/20 0.40
PLD2 O14939 7/20 0.39
PLD1 Q13393 7/20 0.39
USP2 O75604 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
TSHR P16473 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
TNKS O95271 1/20 0.37
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
MEN1 O00255 1/20 0.37
SLC22A2 O15244 1/20 0.37
NR1I2 O75469 1/20 0.37
GMNN O75496 1/20 0.37
LMNA P02545 1/20 0.37
GLA P06280 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1834952 0.89 CALCRL (0.48) CALCRLTNKSPARP1PARP2DRD2
SCHEMBL1837014 0.88 CALCRL (0.48) CALCRLBCHEACHETNKSPARP1
SCHEMBL3403017 0.83 OPRM1 (0.50) PLD2PLD1CYP2D6TSHRBCHE
SCHEMBL1835272 0.83 OPRM1 (0.50) PLD2PLD1CYP2D6TSHRBCHE
SCHEMBL1834571 0.83 NPY5R (0.44) CYP2D6BCHEACHELMNAADRB2
SCHEMBL1832267 0.82 OPRK1 (0.43) PLD2PLD1CYP2D6BCHEACHE
SCHEMBL1832648 0.82 OPRK1 (0.43) PLD2PLD1CYP2D6BCHEACHE
SCHEMBL1840373 0.81 CALCRL (0.42) CALCRLTNKSPARP1PARP2DRD2
SCHEMBL3805948 0.80 CYP2D6 (0.42) PLD2PLD1USP2CYP1A2CYP2D6
SCHEMBL1838176 0.79 OPRK1 (0.50) PLD2PLD1USP2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1997805-A1 Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans Commissariat à l'Energie Atomique (FR) 2008-12-03 EP claimed
EP-2155676-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS Commissariat à l'Energie Atomique (FR) 2010-02-24 EP disclosed
WO-2008146172-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY, APPLICATIONS THEREOF TO THE TREATMENT OF INFECTIOUS DISEASES CAUSED BY APICOMPLEXANS COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-12-04 WO disclosed