SCHEMBL3723967

SCHEMBL3723967

CC(C)(C)OC(=O)NCCN(C(=O)C(=O)O)c1cccc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 1/20 0.55
NQO2 P16083 1/20 0.47
CKS1B P61024 1/20 0.45
SKP1 P63208 1/20 0.45
SKP2 Q13309 1/20 0.45
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
ALDH1A1 P00352 3/20 0.41
IDO1 P14902 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
KDM4A O75164 1/20 0.40
KMT2A Q03164 3/20 0.39
BCHE P06276 1/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MALT1 Q9UDY8 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722147 0.82 DRD2 (0.46) NQO2CKS1BSKP1SKP2IDO1
SCHEMBL3724621 0.79 CKS1B (0.44) NQO2CKS1BSKP1SKP2IDO1
SCHEMBL31393816 0.76 TDP1 (0.45) CKS1BSKP1SKP2ALDH1A1IDO1
SCHEMBL15283620 0.74 CKS1B (0.50) NQO2CKS1BSKP1SKP2CTSS
SCHEMBL29695238 0.74 NQO2 (0.50) NQO2CKS1BSKP1SKP2CTSS
SCHEMBL1579453 0.73 NQO2 (0.75) NQO2CTSSCTSKKDM4A
Hydrochloric Acid SCHEMBL3722949 0.72 MMP9 (0.50) MMP9ALDH1A1L3MBTL1KMT2ARAB9A
SCHEMBL4832420 0.72 KEAP1 (0.44) MMP9CTSSCTSKALDH1A1L3MBTL1
SCHEMBL23649248 0.71 NQO2 (0.65) NQO2CTSSCTSKKDM4A
SCHEMBL15189256 0.71 NPC1 (0.52) CKS1BSKP1SKP2ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125103-A1 DIKETOPIPERAZINE DERIVATIVES AS P2X7 MODULATORS GLAXO GROUP LIMITED (GB) 2010-11-04 WO disclosed