SCHEMBL3797155

SCHEMBL3797155

CCC(=O)Nc1ccc2nc(Oc3ccc(OCC4CC4)cc3C)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.42
RAB9A P51151 2/20 0.39
NOTUM Q6P988 1/20 0.39
NPC1 O15118 1/20 0.39
ACACB O00763 3/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 1/20 0.38
ACACA Q13085 1/20 0.38
HSF1 Q00613 1/20 0.38
PDE4B Q07343 1/20 0.38
MAPT P10636 4/20 0.38
RXFP1 Q9HBX9 3/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPK14 Q16539 1/20 0.37
MCHR1 Q99705 3/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076357 0.84 ACACB (0.47) ACACBCYP3A4CYP2C9ACACA
SCHEMBL3724232 0.84 PDE4B (0.46) ACACBCYP3A4CYP2C9ACACAPDE4B
SCHEMBL3722666 0.81 MAOA (0.37) ACACBCYP3A4CYP2C9ACACAMAPT
SCHEMBL3721926 0.80 PDE4B (0.44) ACACBCYP3A4CYP2C9ACACAPDE4B
SCHEMBL3724233 0.78 ACACB (0.37) ACACBCYP3A4CYP2C9ACACAMCHR1
SCHEMBL13077252 0.78 ACACB (0.46) ACACBCYP3A4CYP2C9ACACA
SCHEMBL3720529 0.76 ACACB (0.37) ACACBCYP3A4CYP2C9ACACAMCHR1
SCHEMBL3718624 0.76 ACACB (0.46) ACACBCYP3A4CYP2C9ACACAMAPT
SCHEMBL3721287 0.75 ACACA (0.51) ACACBCYP3A4CYP2C9ACACA
SCHEMBL3721288 0.75 MTNR1A (0.45) MTNR1AACACBCYP3A4CYP2C9ACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO claimed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed