SCHEMBL3724438

SCHEMBL3724438

CN(C)CCOc1[c]ccc(-c2ccnn2C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP19A1 P11511 1/20 0.42
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ICMT O60725 2/20 0.35
EGLN2 Q96KS0 1/20 0.34
KAT2B Q92831 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PI4KA P42356 1/20 0.34
PIK3CG P48736 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
CHRNB2 P17787 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723622 0.78 ROCK2 (0.42) CYP2D6CYP2C9CYP3A4HRH3CHRNB2
SCHEMBL3805901 0.72 ROCK2 (0.58)
SCHEMBL3715554 0.72 PIM1 (0.46) HRH3
SCHEMBL333569 0.69 PIK3CD (0.41) CYP1A2CYP2D6CYP2C9CYP2C19CYP3A4
SCHEMBL5096842 0.69 MAPT (0.50) KCNH2HRH3CHRNB2CHRNA4ADRA1A
SCHEMBL7387972 0.68 MAPT (0.41) HRH3CHRNB2CHRNA4
SCHEMBL5577859 0.68 HTR2A (0.47) ADRA1AHTR2AHTR2C
SCHEMBL5553179 0.66 KDM4E (0.40) HRH3CHRNB2CHRNA4
SCHEMBL3713952 0.66 ROCK2 (0.51) HRH3
SCHEMBL4360471 0.65 GSR (0.37) HRH3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed