SCHEMBL3715554

SCHEMBL3715554

CN(C)CCOc1[c]ccc(-c2ccnc(N)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 7/20 0.46
PIM3 Q86V86 6/20 0.46
PIM2 Q9P1W9 6/20 0.46
HRH3 Q9Y5N1 2/20 0.42
KMO O15229 1/20 0.41
AURKA O14965 2/20 0.40
CHUK O15111 1/20 0.40
PDPK1 O15530 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CDK2 P24941 1/20 0.40
KDR P35968 1/20 0.40
TGFBR1 P36897 1/20 0.40
SYK P43405 1/20 0.40
JAK3 P52333 1/20 0.40
ROCK1 Q13464 1/20 0.40
AURKB Q96GD4 1/20 0.40
MAP3K5 Q99683 1/20 0.40
HSP90AA1 P07900 1/20 0.39
PRKACA P17612 1/20 0.39
ADORA2A P29274 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225822 0.78 MEN1 (0.54) PIM1PIM3PIM2HRH3AURKA
SCHEMBL3656028 0.78 ROCK2 (0.60) PIM1PIM3PIM2HRH3KMO
SCHEMBL3722649 0.77 HTR7 (0.43) PIM1PIM3PIM2HRH3KMO
SCHEMBL3713494 0.77 CDK2 (0.39) KMOAURKACHUKPDPK1RPS6KB1
SCHEMBL3723622 0.77 ROCK2 (0.42) PIM1HRH3CDK2ROCK1PRKACA
SCHEMBL3805901 0.73 ROCK2 (0.58) ROCK1
SCHEMBL3656027 0.72 CDC7 (0.50) PIM1PIM3PIM2KMOCDK2
SCHEMBL4703487 0.72 MEN1 (0.53) PIM1PIM3PIM2HRH3AURKA
SCHEMBL3724438 0.72 CYP1A2 (0.42) HRH3
SCHEMBL3720566 0.70 KMO (0.43) KMOAURKACHUKPDPK1RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed