SCHEMBL3723622

SCHEMBL3723622

CN(C)CCOc1[c]ccc(-c2ccncc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.42
CDC7 O00311 1/20 0.42
MAP4K4 O95819 1/20 0.42
PIM1 P11309 1/20 0.42
PRKACA P17612 1/20 0.42
CDK2 P24941 1/20 0.42
GSK3B P49841 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
NTRK1 P04629 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
PRKCI P41743 1/20 0.38
BRAF P15056 6/20 0.38
BCHE P06276 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
ROCK1 Q13464 2/20 0.36
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3805901 0.80 ROCK2 (0.58) ROCK2ROCK1
SCHEMBL3724438 0.78 CYP1A2 (0.42) CHRNB2CHRNA4HRH3CYP3A4CYP2D6
SCHEMBL3715554 0.77 PIM1 (0.46) PIM1PRKACACDK2HRH3ROCK1
SCHEMBL5096842 0.74 MAPT (0.50) CHRNB2CHRNA4HRH3
SCHEMBL3725350 0.74 MAPT (0.36) ROCK2CDC7MAP4K4PIM1PRKACA
SCHEMBL4137082 0.73 CYP2D6 (0.66) CHRNB2CHRNA4HRH3BRAFCYP3A4
SCHEMBL3713952 0.73 ROCK2 (0.51) ROCK2PIM1CLK4HRH3ROCK1
SCHEMBL7387972 0.73 MAPT (0.41) CHRNB2CHRNA4HRH3
SCHEMBL20703483 0.72 CHRNB2 (0.50) CHRNB2CHRNA4HRH3CYP2D6CYP2C9
SCHEMBL5553179 0.71 KDM4E (0.40) PIM1CHRNB2CHRNA4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed