SCHEMBL3725838

SCHEMBL3725838

COC(=O)c1cc(-c2cn(Cc3ccccc3)nc2Cl)c(Cl)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
KMT2A Q03164 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RAF1 P04049 1/20 0.42
SCD O00767 3/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ADCY10 Q96PN6 1/20 0.40
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CREBBP Q92793 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC7 Q8WUI4 2/20 0.38
SCD5 Q86SK9 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC2 Q92769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3725017 0.90 SCD (0.39) KDM4EKMT2ASCDALDH1A1POLB
SCHEMBL3724299 0.81 POLQ (0.50) KDM4EKMT2ASMN1; SMN2POLBTDP1
SCHEMBL3724975 0.80 KDM4E (0.45) KDM4EKMT2ASMN1; SMN2RAF1SCD
SCHEMBL13260110 0.78 KDM4E (0.43) KDM4EKMT2ASMN1; SMN2RAF1SCD
SCHEMBL3725282 0.76 KMT2A (0.41) KDM4EKMT2ASMN1; SMN2RAF1SCD
SCHEMBL3721607 0.75 KDM4E (0.43) KDM4EKMT2ASMN1; SMN2RAF1SCD
SCHEMBL3724448 0.75 POLQ (0.41) KDM4EKMT2ASMN1; SMN2RAF1SCD
SCHEMBL3722206 0.72 POLQ (0.52) KDM4EKMT2ASMN1; SMN2CREBBP
SCHEMBL3724391 0.72 HDAC1 (0.42) KDM4EKMT2ASMN1; SMN2RAF1SCD
SCHEMBL17398413 0.71 HSP90AA1 (0.48) KDM4EKMT2ASMN1; SMN2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093885-A1 INHIBITORS OF AKT ACTIVITY GLAXOSMITHKLINE LLC (US) 2010-08-19 WO disclosed
WO-2010093885-A1 INHIBITORS OF AKT ACTIVITY GLAXOSMITHKLINE LLC (US) 2010-08-19 WO disclosed