SCHEMBL3725282

SCHEMBL3725282

C=Cc1nn(Cc2ccccc2)cc1-c1cc(C(=O)OC)sc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
RAF1 P04049 1/20 0.39
ALDH1A1 P00352 4/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 1/20 0.37
SCD O00767 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724448 0.87 POLQ (0.41) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL3724975 0.86 KDM4E (0.45) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL13260110 0.85 KDM4E (0.43) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL3722206 0.79 POLQ (0.52) KMT2AKDM4ESMN1; SMN2POLQ
SCHEMBL3724391 0.77 HDAC1 (0.42) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL3725838 0.76 KDM4E (0.45) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL3725819 0.76 HDAC1 (0.42) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL3721607 0.73 KDM4E (0.43) KMT2AKDM4ESMN1; SMN2HDAC1HDAC7
SCHEMBL3724299 0.71 POLQ (0.50) KMT2AKDM4ESMN1; SMN2POLBTDP1
SCHEMBL13260970 0.69 POLQ (0.48) KMT2AKDM4ESMN1; SMN2HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093885-A1 INHIBITORS OF AKT ACTIVITY GLAXOSMITHKLINE LLC (US) 2010-08-19 WO disclosed
WO-2010093885-A1 INHIBITORS OF AKT ACTIVITY GLAXOSMITHKLINE LLC (US) 2010-08-19 WO disclosed