SCHEMBL3726439

SCHEMBL3726439

CCOc1ccc(Oc2ccc3cc(C(C)Nc4ccon4)ccc3c2)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 5/20 0.39
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
HTR2A P28223 3/20 0.34
SLC6A4 P31645 3/20 0.34
KCNH2 Q12809 3/20 0.34
PARG Q86W56 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
ACACA Q13085 1/20 0.33
FFAR1 O14842 1/20 0.33
P2RX3 P56373 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
CRHR1 P34998 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726441 0.80 RAB9A (0.38) ACACBRAB9AKDM4EMAPTPARG
SCHEMBL13077221 0.76 ACACB (0.57) ACACBAKR1C3AKR1C2ACACA
SCHEMBL3716937 0.76 AKR1C3 (0.51) ACACBAKR1C3AKR1C2MAPTPARG
SCHEMBL3721758 0.70 KDM4E (0.37) ACACBAKR1C3AKR1C2KDM4EMAPT
SCHEMBL13077068 0.69 ACACB (0.56) ACACBAKR1C3AKR1C2ACACA
SCHEMBL3721938 0.69 ACACB (0.59) ACACBACACA
SCHEMBL3716764 0.67 ACACB (0.54) ACACBACACA
SCHEMBL3723075 0.67 ACACB (0.57) ACACBACACA
SCHEMBL3726992 0.67 ESRRA (0.53) ACACBAKR1C3AKR1C2KDM4EMAPT
SCHEMBL1390808 0.66 RAB9A (0.41) ACACBRAB9AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO claimed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed