SCHEMBL3721758

SCHEMBL3721758

CCOc1ccc(Oc2ccc3cc(C(C)N(c4ccon4)S(=O)(=O)c4ccc([N+](=O)[O-])cc4)ccc3c2)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 3/20 0.36
PTPN1 P18031 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
CYP26A1 O43174 1/20 0.34
CYP3A4 P08684 1/20 0.34
PDE7A Q13946 1/20 0.33
TBXA2R P21731 2/20 0.33
MAPT P10636 3/20 0.33
KMT2A Q03164 3/20 0.33
NPSR1 Q6W5P4 2/20 0.33
LMNA P02545 1/20 0.33
PTGS2 P35354 1/20 0.33
MEN1 O00255 2/20 0.32
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721759 0.82 KDM4E (0.37) KDM4EALDH1A1PTPN1PDE7ATBXA2R
SCHEMBL1390796 0.74 MEN1 (0.35) ALDH1A1PTPN1MAPTKMT2ANPSR1
SCHEMBL3726439 0.70 ACACB (0.39) KDM4EMAPTKMT2AMEN1ACACB
SCHEMBL3716937 0.67 AKR1C3 (0.51) MAPTKMT2AMEN1ACACBAKR1C3
SCHEMBL13077221 0.63 ACACB (0.57) LMNAACACBAKR1C3AKR1C2
SCHEMBL22069593 0.62 PDE7A (0.74) KDM4EALDH1A1CYP3A4PDE7AMAPT
SCHEMBL27708666 0.62 PTGS2 (0.57) KDM4EALDH1A1CYP3A4PDE7ATBXA2R
SCHEMBL3726441 0.62 RAB9A (0.38) KDM4EMAPTACACB
SCHEMBL23014061 0.61 ALDH1A1 (0.45) KDM4EALDH1A1PSEN1PSEN2APH1B
SCHEMBL11163357 0.60 ALDH1A1 (0.54) KDM4EALDH1A1PDE7AMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed