SCHEMBL3728167

SCHEMBL3728167

CCCCCc1ccc2c3cc(C=Cc4cccc(F)c4)ccc3n(S(=O)(=O)c3ccccc3)c2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.37
PTGDR Q13258 2/20 0.37
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
FLT3 P36888 2/20 0.35
ALDH1A2 O94788 1/20 0.34
ALDH1A1 P00352 1/20 0.34
NFE2L2 Q16236 1/20 0.34
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
PARP1 P09874 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724852 0.93 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3724854 0.93 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL676108 0.82 HTR2A (0.43) PTGDR2PTGDRALDH1A2ALDH1A1NFE2L2
SCHEMBL3726812 0.82 PTGDR2 (0.36) PTGDR2PTGDRPSEN1PSEN2APH1B
SCHEMBL675181 0.82 NFE2L2 (0.40) PTGDR2PTGDRALDH1A2ALDH1A1NFE2L2
SCHEMBL3726800 0.81 HTR6 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3728168 0.76 PSEN1 (0.36) PTGDR2PTGDRPSEN1PSEN2APH1B
SCHEMBL676120 0.76 HTR6 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3721458 0.76 CNR2 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3721754 0.75 ALDH1A1 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed