SCHEMBL3728532

SCHEMBL3728532

COc1cc(C(C#N)C(=O)C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
RAPGEF3 O95398 1/20 0.36
RAPGEF4 Q8WZA2 1/20 0.36
TMPRSS4 Q9NRS4 2/20 0.36
EPHX2 P34913 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADCY8 P40145 2/20 0.35
ADCY1 Q08828 2/20 0.35
P2RX1 P51575 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL943020 1.00 RXRA (0.40) RXRARXRBRXRGHDAC3HDAC1
SCHEMBL10850841 0.83 RXRA (0.40) RXRARXRBRXRGHDAC3HDAC1
SCHEMBL1008766 0.79 RAPGEF3 (0.40) HDAC3HDAC1HDAC2HDAC6RAPGEF3
SCHEMBL10776182 0.78 RXRA (0.49) RXRARXRBRXRGKMT2AMEN1
SCHEMBL586419 0.73 AKR1C3 (0.54) RXRARXRBRXRGHDAC3HDAC1
SCHEMBL10851034 0.72 SMN1; SMN2 (0.38) RAPGEF3RAPGEF4KMT2AMEN1SMN1; SMN2
SCHEMBL1056618 0.72 CYP1A2 (0.48) KMT2ALMNAHTTKDM4E
SCHEMBL585795 0.71 RXRA (0.43) RXRARXRBRXRGHDAC3HDAC1
SCHEMBL10084735 0.71 RXRA (0.40) RXRARXRBRXRGHDAC3HDAC1
SCHEMBL7271607 0.70 GRN (0.35) RAPGEF3RAPGEF4AKR1C3AKR1C2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010136145-A1 PYRAZINYLPYRAZOLES BAYER CROPSCIENCE AG (DE) 2010-12-02 WO disclosed