SCHEMBL3728544

SCHEMBL3728544

CCCCCc1ccc2c3cc(-c4ccc(CN5CCOCC5)cc4)ccc3n(S(=O)(=O)c3ccccc3)c2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ATM Q13315 1/20 0.42
ALDH1A1 P00352 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PIK3CD O00329 1/20 0.39
MTOR P42345 1/20 0.39
TSHR P16473 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
CHEK1 O14757 2/20 0.38
ICMT O60725 1/20 0.38
HDAC1 Q13547 1/20 0.38
JAK2 O60674 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726800 0.86 HTR6 (0.40) ICMTPSEN1PSEN2APH1BNCSTN
SCHEMBL3668206 0.85 PARP1 (0.45) NPC1RAB9AATMALDH1A1NPSR1
SCHEMBL676293 0.85 NPC1 (0.45) NPC1RAB9AATMALDH1A1NPSR1
SCHEMBL3724235 0.83 PIK3CD (0.40) NPC1RAB9AATMPIK3CDMTOR
SCHEMBL3723156 0.82 NOD2 (0.37) NPC1RAB9AALDH1A1PIK3CDMTOR
SCHEMBL676120 0.81 HTR6 (0.44) RAB9AALDH1A1TSHRPSEN1PSEN2
SCHEMBL3721458 0.79 CNR2 (0.37) ALDH1A1TSHRPSEN1PSEN2APH1B
SCHEMBL677027 0.77 PIK3CD (0.47) NPC1RAB9AATMALDH1A1NPSR1
SCHEMBL3721754 0.77 ALDH1A1 (0.40) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL3666429 0.76 PIK3CA (0.44) NPC1RAB9AATMALDH1A1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed