SCHEMBL3728883

SCHEMBL3728883

COc1c[c]ccc1-c1nc(Br)c[nH]1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DCUN1D1 Q96GG9 2/20 0.31
AMY1A P0DUB6 3/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2445492 0.84 DCUN1D1 (0.32) DCUN1D1ALDH1A1GAA
SCHEMBL3637473 0.73 IMPDH2 (0.43) ALDH1A1GAA
SCHEMBL6541679 0.73 CA1 (0.38) ALDH1A1
SCHEMBL3733422 0.69 PDE5A (0.31)
SCHEMBL3722110 0.68 ROCK2 (0.40)
SCHEMBL4267696 0.68
SCHEMBL2039605 0.67 FYN (0.40)
SCHEMBL2041601 0.67 CYP2A6 (0.48)
SCHEMBL28789059 0.67 ERN1 (0.42) ALDH1A1
SCHEMBL230060 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed