SCHEMBL3729968

SCHEMBL3729968

CC(C)(C)OC(=O)Nc1cccc2cc(N)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
PLAU P00749 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CASP6 P55212 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
TRPV1 Q8NER1 2/20 0.41
MAPK14 Q16539 2/20 0.40
SRC P12931 1/20 0.40
MAPK9 P45984 1/20 0.40
DDR2 Q16832 1/20 0.40
NQO2 P16083 1/20 0.39
BRD9 Q9H8M2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
MMP8 P22894 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6101638 0.85 NQO2 (0.51) ALDH1A1HPGDRXFP1CASP6KDM4E
SCHEMBL27453735 0.84 RXFP1 (0.46) ALDH1A1HPGDPLAURXFP1CASP6
SCHEMBL30077817 0.84 RXFP1 (0.46) ALDH1A1HPGDPLAURXFP1CASP6
SCHEMBL2396852 0.83 ALDH1A1 (0.63) ALDH1A1HPGDKDM4EGAAMAPK14
SCHEMBL14059000 0.81 CASP6 (0.68) ALDH1A1HPGDRXFP1CASP6KDM4E
SCHEMBL3246360 0.78 TRPV1 (0.63) ALDH1A1KDM4ETRPV1
SCHEMBL421016 0.78 MAPK14 (0.47) ALDH1A1HPGDPLAURXFP1KDM4E
SCHEMBL115453 0.77 RXFP1 (0.43) ALDH1A1HPGDRXFP1CASP6TRPV1
SCHEMBL15160030 0.77 GAA (0.52) RXFP1GAANPC1
SCHEMBL2227781 0.77 AAK1 (0.48) RXFP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152664-A1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS Brystol-Myers Squibb Company (US) 2010-02-17 EP disclosed
WO-2008157162-A1 DIPEPTIDE ANALOGS AS COAGULATION FACTOR INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-24 WO disclosed