SCHEMBL3735283

SCHEMBL3735283

CC(=O)NC(NC(C)=O)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.63
ALDH1A1 P00352 4/20 0.59
CNR2 P34972 3/20 0.57
TSHR P16473 1/20 0.53
SRC P12931 1/20 0.52
MTNR1A P48039 3/20 0.52
MTNR1B P49286 3/20 0.52
CNR1 P21554 1/20 0.49
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 2/20 0.48
NAPRT Q6XQN6 1/20 0.48
CYP2C19 P33261 1/20 0.47
KDM4E B2RXH2 1/20 0.47
CTRB1 P17538 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5307928 0.94 CYP1A2 (0.57) CYP1A2ALDH1A1CNR2TSHRSRC
SCHEMBL13392839 0.89 CYP1A2 (0.52) CYP1A2ALDH1A1CNR2TSHRSRC
SCHEMBL4196370 0.87 CYP1A2 (0.50) CYP1A2ALDH1A1CNR2TSHRSRC
SCHEMBL6675601 0.87 CYP1A2 (0.50) CYP1A2ALDH1A1CNR2TSHRSRC
SCHEMBL3742027 0.85 CNR2 (0.57) CYP1A2ALDH1A1CNR2TSHRMTNR1A
SCHEMBL3729174 0.85 CNR2 (0.57) CYP1A2ALDH1A1CNR2TSHRMTNR1A
SCHEMBL425361 0.84 ALDH1A1 (0.58) ALDH1A1TSHRSRCMTNR1AMTNR1B
SCHEMBL9777891 0.83 CNR2 (0.59) ALDH1A1CNR2SRCCNR1KMT2A
SCHEMBL640385 0.82 ACACB (0.65) ALDH1A1POLBKMT2AHSD17B10KDM4E
SCHEMBL6693251 0.82 MTNR1A (0.48) CYP1A2ALDH1A1SRCMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100278730-A1 Non-Invasive Molecular Imaging of Cellular Histone Deacetylase Substrate Using Magnetic Resonance Spectroscopy (MRS) or Positron Emission Tomography (PET) BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2010-11-04 US claimed
WO-2009009179-A2 NON-INVASIVE MOLECULAR IMAGING OF CELLULAR HISTONE DEACETYLASE SUBSTRATE USING MAGNETIC RESONANCE SPECTROSCOPY (MRS) OR POSITRON EMISSION TOMOGRAPHY (PET) BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2009-01-15 WO claimed
US-20100278730-A1 Non-Invasive Molecular Imaging of Cellular Histone Deacetylase Substrate Using Magnetic Resonance Spectroscopy (MRS) or Positron Emission Tomography (PET) BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2010-11-04 US disclosed
WO-2009009179-A2 NON-INVASIVE MOLECULAR IMAGING OF CELLULAR HISTONE DEACETYLASE SUBSTRATE USING MAGNETIC RESONANCE SPECTROSCOPY (MRS) OR POSITRON EMISSION TOMOGRAPHY (PET) BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2009-01-15 WO disclosed
US-4083868-A INTRAOCULAR PRESSURE LOWERING AGENTS ABBOTT LABORATORIES (US) 1978-04-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100278730-A1 Non-Invasive Molecular Imaging of Cellular Histone Deacetylase Substrate Using Magnetic Resonance Spectroscopy (MRS) or Positron Emission Tomography (PET) HDAC1, HDAC3, HDAC10 CYP1A2 4709/4885ALDH1A1 2246/4885CNR2 4288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.