SCHEMBL3759003

SCHEMBL3759003

NC(C(=O)N1CCC1)c1ccccc1-c1[c]nccc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP7 Q9UHL4 9/20 0.39
DPP4 P27487 8/20 0.39
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
PREP P48147 1/20 0.31
PTAFR P25105 1/20 0.31
TSHR P16473 2/20 0.30
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HRH1 P35367 1/20 0.30
ROCK2 O75116 1/20 0.30
CYP3A4 P08684 1/20 0.30
RECQL P46063 1/20 0.30
CHRM3 P20309 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3761660 0.98 DPP7 (0.41) DPP7DPP4ALDH1A1HTTPREP
SCHEMBL4003839 0.79 ALDH1A1 (0.40) DPP7DPP4ALDH1A1HTTPTAFR
SCHEMBL3760379 0.77 TSHR (0.54) ALDH1A1HTTTSHRSMN1; SMN2RECQL
SCHEMBL3759224 0.76 CTSK (0.34)
SCHEMBL3759087 0.76 KCNA5 (0.33) ALDH1A1HTTSMN1; SMN2CYP3A4
SCHEMBL3765034 0.75 HTR2C (0.35) DPP7DPP4ALDH1A1HTTTSHR
SCHEMBL3756110 0.74 KCNA5 (0.35) CYP3A4
SCHEMBL3754962 0.74 LMNA (0.47) ALDH1A1TSHRSMN1; SMN2CHRM3CHRM1
SCHEMBL3760644 0.74 TSHR (0.57) ALDH1A1HTTTSHRNPC1RAB9A
SCHEMBL3756633 0.74 CTSL (0.35) DPP7DPP4ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029570-B1 FUSED THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA SA (BE) 2014-10-15 EP disclosed
US-8324204-B2 Fused thiophene derivatives as kinase inhibitors UCB PHARMA SA (BE) 2012-12-04 US disclosed
US-20100305066-A1 Fused Thiophene Derivatives as Kinase Inhibitors UCB PHARMA S.A. (BE) 2010-12-02 US disclosed
WO-2009122148-A1 FUSED THIOPHENE AND THIAZOLE DERIVATIVES AS PI3K KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-10-08 WO disclosed
WO-2009071895-A1 FUSED THIAZOLE AND THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
WO-2009071890-A1 TRICYCLIC KINASE INHIBITORS UCB PHARMA S.A. (BE) 2009-06-11 WO disclosed
EP-2029570-A1 FUSED THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB Pharma S.A. (BE) 2009-03-04 EP disclosed
WO-2007141504-A1 FUSED THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2007-12-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100305066-A1 Fused Thiophene Derivatives as Kinase Inhibitors PIKFYVE, PI4KA, PIK3CA DPP7 421/4885DPP4 462/4885ALDH1A1 3061/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.