SCHEMBL3761271

SCHEMBL3761271

CCOc1ncncc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.38
ALDH1A1 P00352 2/20 0.36
CYP17A1 P05093 1/20 0.36
TDP1 Q9NUW8 2/20 0.34
TSHR P16473 1/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
MAPT P10636 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CA12 O43570 2/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735866 0.78
SCHEMBL31008552 0.78
SCHEMBL23143263 0.76 AOC3 (0.44) AOC3CYP17A1KDM4EHPGDSMN1; SMN2
SCHEMBL22339621 0.75 CYP17A1 (0.36) AOC3ALDH1A1CYP17A1TDP1MAPT
SCHEMBL22574812 0.75 HPGD (0.40) AOC3ALDH1A1CYP17A1TSHRMEN1
SCHEMBL21725546 0.75 CYP17A1 (0.36) AOC3CYP17A1MEN1KMT2AMAPT
SCHEMBL10273189 0.75 CYP17A1 (0.39) AOC3CYP17A1MEN1KMT2AKDM4E
SCHEMBL13363832 0.75 CYP17A1 (0.39) AOC3ALDH1A1CYP17A1MEN1KMT2A
SCHEMBL16702537 0.75 ALDH1A1 (0.44) ALDH1A1CYP17A1MEN1KMT2AMAPT
SCHEMBL21725547 0.73 AOC3 (0.37) AOC3CYP17A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116924976-A Diaryl heterocyclic amine compound, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2023-10-24 CN disclosed
CN-110225912-B GSK-3 inhibitors 百时美施贵宝公司 2022-10-21 CN disclosed
EP-3544980-B1 GSK-3 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
EP-3544980-B1 GSK-3 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
US-10774086-B2 GSK-3 inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2020-09-15 US disclosed
EP-3544980-A1 GSK-3 INHIBITORS Bristol-Myers Squibb Company (US) 2019-10-02 EP disclosed
US-20190276463-A1 GSK-3 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2019-09-12 US disclosed
WO-2018098411-A1 GSK-3 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-31 WO disclosed
WO-2018098411-A1 GSK-3 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-31 WO disclosed
US-7851473-B2 Amide compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-14 US disclosed
US-20080312226-A1 Amide Compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-12-18 US disclosed
EP-1813606-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-08-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080312226-A1 Amide Compound FAAH, FAAH2, CNR2 AOC3 371/4885ALDH1A1 353/4885CYP17A1 2277/4885
US-20190276463-A1 GSK-3 INHIBITORS GSK3B, GSK3A, GSKIP AOC3 3685/4885ALDH1A1 4339/4885CYP17A1 134/4885
US-10774086-B2 GSK-3 inhibitors GSK3B, GSK3A, GSKIP AOC3 3685/4885ALDH1A1 4339/4885CYP17A1 134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.