SCHEMBL3767589

SCHEMBL3767589

N#CCCc1ccc(C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
RARB P10826 6/20 0.49
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
MAPT P10636 2/20 0.46
RARA P10276 1/20 0.46
MTOR P42345 1/20 0.46
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45
SRD5A2 P31213 2/20 0.43
PPARA Q07869 1/20 0.42
MMP9 P14780 1/20 0.42
MMP13 P45452 1/20 0.42
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6480448 0.89 RARB (0.54) ALDH1A1RARBTP53TSHRKMT2A
SCHEMBL3455668 0.82 PLA2G10 (0.48) ALDH1A1TSHRKMT2AMEN1MAPT
SCHEMBL4946030 0.82 KMT2A (0.55) ALDH1A1KMT2AMEN1MAPTNR1H2
SCHEMBL11580792 0.82 MEN1 (0.44) ALDH1A1KMT2AMEN1MAPTNR1H2
SCHEMBL4968695 0.82 ALDH1A1 (0.52) ALDH1A1RARBTP53TSHRKMT2A
Terephthalic Acid SCHEMBL4612225 0.80 TSHR (0.67) ALDH1A1RARBTP53TSHRKMT2A
SCHEMBL70166 0.80 TSHR (0.67) ALDH1A1RARBTP53TSHRKMT2A
SCHEMBL31747387 0.80 ALDH1A1 (0.50) ALDH1A1RARBTP53TSHRKMT2A
SCHEMBL8764230 0.80 MEN1 (0.64) ALDH1A1TSHRKMT2AMEN1NR1H2
SCHEMBL211305 0.79 ALDH1A1 (0.54) ALDH1A1RARBTP53TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102123987-A Cycloalkylidene and heterocycloalkylidene histone deacetylase inhibitor compounds GILEAD COLORADO INC 2011-07-13 CN disclosed
US-7851658-B2 Palladium-catalyzed carbon-carbon bond forming reactions PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-12-14 US disclosed
WO-2007008226-A9 PALLADIUM-CATALYZED CARBON-CARBON BOND FORMING REACTIONS HARVARD COLLEGE (US) 2007-05-24 WO disclosed
US-20070066851-A1 Palladium-catalyzed carbon-carbon bond forming reactions NAVY, SECRETARY OF THE UNITED STATES OF AMERICA 2007-03-22 US disclosed
WO-2007008226-A2 PALLADIUM-CATALYZED CARBON-CARBON BOND FORMING REACTIONS THE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2007-01-18 WO disclosed
US-20050075345-A1 Novel inhibitor compounds specific of secreted non-pancreatic human a<sb>2</sb>phospholipase of group II YANG JI CHEMICAL COMPANY LTD. (KR) 2005-04-07 US disclosed
US-5145854-A 1-formyl-5,8,10-trideazafolates NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 1992-09-08 US disclosed
US-4105653-A HETERYL-AZO-PHENYL DISPERSE DYESTUFFS CONTAINING A Z-SUBSTITUTED BENZOLYLOXYALKYL RADICAL, WHEREIN Z IS 2-CYANOVINYL 2-CYANOETHYL OR 2-CHLORO-2-CYANOETHYL PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1978-08-08 US disclosed
US-3987027-A DISPERSE AZO DYES PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1976-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070066851-A1 Palladium-catalyzed carbon-carbon bond forming reactions APEX1, PCNA, DNMT3A ALDH1A1 564/4885RARB 3349/4885TP53 2229/4885
US-20050075345-A1 Novel inhibitor compounds specific of secreted non-pancreatic human a<sb>2</sb>phospholipase of group II AMY2A, PNLIP, IAPP ALDH1A1 3782/4885RARB 2571/4885TP53 3676/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.