Iodixanol

Iodixanol

SCHEMBL37712

CC(=O)N(CC(O)CN(C(C)=O)c1c(I)c(C(=O)NC[C@H](O)CO)c(I)c(C(=O)NC[C@H](O)CO)c1I)c1c(I)c(C(=O)NC[C@H](O)CO)c(I)c(C(=O)NC[C@H](O)CO)c1I

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 1.00
CYP2C19 P33261 1/20 0.95
HIF1A Q16665 1/20 0.95
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
MAP2K1 Q02750 7/20 0.33
MAP2K2 P36507 2/20 0.32
PRKCZ Q05513 1/20 0.32
IARS2 Q9NSE4 1/20 0.32
CYP2C9 P11712 1/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodixanol SCHEMBL8845042 1.00 LMNA (1.00) LMNACYP2C19HIF1AEGFRSRC
Iodixanol SCHEMBL21546 1.00 LMNA (1.00) LMNACYP2C19HIF1AEGFRSRC
Iodixanol SCHEMBL22645199 0.99 LMNA (0.97) LMNACYP2C19HIF1AEGFRSRC
Iohexol SCHEMBL8844889 0.97 CYP2C19 (1.00) LMNACYP2C19HIF1AEGFRSRC
Iohexol SCHEMBL31722694 0.97 CYP2C19 (1.00) LMNACYP2C19HIF1AEGFRSRC
Iohexol SCHEMBL37920 0.97 CYP2C19 (1.00) LMNACYP2C19HIF1AEGFRSRC
Iohexol SCHEMBL26501 0.97 CYP2C19 (1.00) LMNACYP2C19HIF1AEGFRSRC
SCHEMBL12589793 0.96 LMNA (0.93) LMNACYP2C19HIF1AEGFRSRC
Iohexol SCHEMBL8711982 0.96 CYP2C19 (0.97) LMNACYP2C19HIF1AEGFRSRC
Iohexol SCHEMBL22719758 0.95 CYP2C19 (0.95) LMNACYP2C19HIF1AEGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2380 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4704924-A1 RADIONUCLIDE-LOADED NANOPARTICLES FOR FOCAL TISSUE ABLATION TRANSLATIONAL AND FUNDAMENTAL TECHNOLOGIES INSTITUTE LLC (US) 2026-03-11 EP claimed
EP-3893913-B1 TRANSFERRIN RECEPTOR TARGETING PEPTIDES FRED HUTCHINSON CANCER CENTER (US) 2025-03-26 EP claimed
US-20250043251-A1 METHOD FOR FURTHER UPSCALING THE LARGE-SCALE PRODUCTION OF THE ONCOLYTIC H-1 PROTOPARVOVIRUS (H-1PV) USING A CARRIER-BASED PRODUCTION PROCESS COMBINED WITH AN OPTIMIZED CELL CULTURE MEDIUM DEUTSCHES KREBSFORSCHUNGSZENTRUM STIFTUNG DES OEFFENTLICHEN RECHTS (DE) 2025-02-06 US claimed
US-20240390364-A1 Novel Pyridine Compositions and their use in methods for preventing or treating diseases, disorders and conditions REID CHRISTOPHER BRIAN (US) 2024-11-28 US claimed
WO-2024226199-A1 RADIONUCLIDE-LOADED NANOPARTICLES FOR FOCAL TISSUE ABLATION RAIKA MEDICAL IMAGING INC. (US) 2024-10-31 WO claimed
US-20240350684-A1 RADIONUCLIDE-LOADED NANOPARTICLES FOR FOCAL TISSUE ABLATION TRANSLATIONAL AND FUNDAMENTAL TECHNOLOGIES INSTITUTE LLC 2024-10-24 US claimed
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO claimed
EP-4408985-A1 METHOD FOR FURTHER UPSCALING THE LARGE-SCALE PRODUCTION OF THE ONCOLYTIC H-1 PROTOPARVOVIRUS (H-1PV) USING A CARRIER-BASED PRODUCTION PROCESS COMBINED WITH AN OPTIMIZED CELL CULTURE MEDIUM Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2024-08-07 EP claimed
WO-2023052429-A1 METHOD FOR FURTHER UPSCALING THE LARGE-SCALE PRODUCTION OF THE ONCOLYTIC H-1 PROTOPARVOVIRUS (H-1PV) USING A CARRIER-BASED PRODUCTION PROCESS COMBINED WITH AN OPTIMIZED CELL CULTURE MEDIUM Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2023-04-06 WO claimed
US-20220169992-A1 OPTIMIZED PARVOVIRUS H-1 PRODUCTION DEUTSCHES KREBSFORSCHUNGSZENTRUM STIFTUNG DES OFFENTLICHEN RECHTS (DE) 2022-06-02 US claimed
CN-1161324-C Yellow polymorphic forms of 5-amino-2, 4, 6-triiodo-N, N' -bis (2, 3-dihydroxypropyl) isophthalamide ��Īɳķ������˾ 2004-08-11 CN claimed
CN-1494435-A Preparation for preventing restenosis �����ڶ���ϣ 2004-05-05 CN claimed
EP-1372737-A2 PREPARATION FOR THE PROPHYLAXIS OF RESTENOSIS Speck, Ulrich (DE) 2004-01-02 EP claimed
CN-1129566-C Method for crystallization of sterically hindered compounds NYCOMBED IMAGING AS (NO) 2003-12-03 CN claimed
CN-1092182-C Process for preparation of contrast agent NYCOMED IMAGING AS (NO) 2002-10-09 CN claimed
WO-2002076509-A2 PREPARATION FOR THE PROPHYLAXIS OF RESTENOSIS SPECK ULRICH (DE) 2002-10-03 WO claimed
CN-1340042-A Preparation of iodixanol NYCOMED IMAGING AS (NO) 2002-03-13 CN claimed
CN-1273574-A Process for crystallisation of sterically hindered compound NYCOMBED IMAGING AS (NO) 2000-11-15 CN claimed
CN-1257479-A Yellow polymorph of 5-amino-2,4,6-triiodo-N,N'-bis(2,3-dihydroxypropyl)-isophthalamide NYCOMED IMAGING AS (NO) 2000-06-21 CN claimed
CN-1228762-A Process for preparation of contrast agent NYCOMED IMAGING AS (NO) 1999-09-15 CN claimed