SCHEMBL3780103

SCHEMBL3780103

CN(C)C(=O)C(Cc1c[nH]c2ccccc12)NC(=O)O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 2/20 0.77
MMP8 P22894 2/20 0.77
MMP14 P50281 1/20 0.77
TACR1 P25103 2/20 0.65
MMP2 P08253 1/20 0.63
ALOX15 P16050 1/20 0.60
ITGB2 P05107 2/20 0.60
ICAM1 P05362 2/20 0.60
ITGAL P20701 2/20 0.60
ACE P12821 3/20 0.59
POLB P06746 2/20 0.56
MAPT P10636 2/20 0.56
KDM4E B2RXH2 1/20 0.56
APAF1 O14727 1/20 0.56
RECQL P46063 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
CCKBR P32239 1/20 0.55
ALDH1A1 P00352 1/20 0.55
HPGD P15428 1/20 0.55
ECE1 P42892 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26647227 0.88 MMP9 (0.61) MMP9MMP8MMP14TACR1ALOX15
SCHEMBL26647233 0.88 MMP9 (0.61) MMP9MMP8MMP14TACR1ALOX15
SCHEMBL8200367 0.87 TACR1 (0.86) MMP9MMP8MMP14TACR1ALOX15
SCHEMBL8200364 0.87 TACR1 (0.86) MMP9MMP8MMP14TACR1ALOX15
SCHEMBL3857226 0.85 ALOX15 (0.74) ALOX15ITGB2ICAM1ITGALACE
SCHEMBL3857229 0.85 ALOX15 (0.74) ALOX15ITGB2ICAM1ITGALACE
SCHEMBL22059460 0.84 MMP9 (0.68) MMP9MMP8MMP14TACR1MMP2
SCHEMBL22059492 0.84 MMP9 (0.68) MMP9MMP8MMP14TACR1MMP2
SCHEMBL25001444 0.84 CTSL (0.68) MMP9MMP8MMP14TACR1MMP2
SCHEMBL3787557 0.84 MMP9 (0.72) MMP9MMP8MMP14MMP2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2260022-B1 SUBSTITUTED CYCLOHEXYLDIAMINES GRUENENTHAL GMBH (DE) 2017-01-04 EP disclosed
EP-2260022-A1 SUBSTITUTED CYCLOHEXYLDIAMINES Grünenthal GmbH (DE) 2010-12-15 EP disclosed
WO-2009118174-A1 SUBSTITUTED CYCLOHEXYLDIAMINES Grünenthal GmbH (DE) 2009-10-01 WO disclosed