SCHEMBL3783787

SCHEMBL3783787

CN(Cl)c1ncccc1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
HPGD P15428 6/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP11B2 P19099 1/20 0.39
POLB P06746 1/20 0.39
LRRK2 Q5S007 1/20 0.39
KCNMA1 Q12791 1/20 0.38
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 2/20 0.36
TSHR P16473 1/20 0.36
ELANE P08246 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6191221 0.85 HTT (0.45) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL21614128 0.80 ALDH1A1 (0.39) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL16580958 0.79 HPGD (0.40) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL12125020 0.79 HPGD (0.43) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL3782096 0.77 HPGD (0.40) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL5200518 0.76 KCNMA1 (0.47) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL1230919 0.76 PTK2 (0.50) ALDH1A1JAK2JAK3HTT
SCHEMBL5584219 0.76 CHRM5 (0.38) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL14068342 0.75 ALDH1A1 (0.35) ALDH1A1HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL3288220 0.74 KDM4E (0.51) ALDH1A1HPGDSMN1; SMN2RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2187893-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2010-05-26 EP disclosed
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed