SCHEMBL378738

SCHEMBL378738

O=C(NCCc1ccccc1)C1(c2ccccc2)CCNCC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.58
CHRM5 P08912 1/20 0.57
CHRM3 P20309 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.56
HTT P42858 1/20 0.56
OPRM1 P35372 1/20 0.50
HDAC1 Q13547 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C19 P33261 1/20 0.50
LMNA P02545 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
EPHX1 P07099 1/20 0.48
MC4R P32245 1/20 0.46
ALDH1A1 P00352 1/20 0.45
CA12 O43570 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
ERCC1 P07992 1/20 0.45
ERCC4 Q92889 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378386 0.92 TACR1 (0.57) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL378422 0.92 TACR1 (0.56) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL2467338 0.89 CHRM5 (0.74) TACR1CHRM5CHRM3SMN1; SMN2L3MBTL1
SCHEMBL476243 0.86 TACR1 (0.71) TACR1SMN1; SMN2HTTOPRM1HDAC1
SCHEMBL378420 0.85 TACR1 (0.48) TACR1CHRM5CHRM3SMN1; SMN2LMNA
SCHEMBL6375805 0.84 SMN1; SMN2 (0.57) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL6543304 0.82 OPRM1 (0.56) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL6623954 0.82 EPHX1 (0.49) TACR1CYP3A4CYP2C19EPHX1MC4R
SCHEMBL2472385 0.81 OPRM1 (0.54) TACR1CHRM5CHRM3SMN1; SMN2HTT
SCHEMBL4965067 0.81 PLAAT3 (0.57) CHRM5CHRM3SMN1; SMN2HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed