SCHEMBL378420

SCHEMBL378420

O=C(NCCc1ccc(F)cc1)C1(c2ccc(F)cc2)CCNCC1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.48
HPGD P15428 1/20 0.46
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
CHRM5 P08912 1/20 0.45
CHRM3 P20309 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
PLAAT3 P53816 1/20 0.43
PLAAT5 Q96KN8 1/20 0.43
PLAAT2 Q9NWW9 1/20 0.43
PLAAT4 Q9UL19 1/20 0.43
POLB P06746 1/20 0.42
CNR1 P21554 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378386 0.94 TACR1 (0.57) TACR1NPC1RAB9ASMN1; SMN2CHRM5
SCHEMBL378738 0.85 TACR1 (0.58) TACR1SMN1; SMN2CHRM5CHRM3ALDH1A1
SCHEMBL5349607 0.81 HDAC4 (0.55) SMN1; SMN2ALDH1A1CNR1LMNA
SCHEMBL10254952 0.80 TACR1 (0.69) TACR1NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL2467338 0.78 CHRM5 (0.74) TACR1NPC1RAB9ASMN1; SMN2CHRM5
SCHEMBL378422 0.77 TACR1 (0.56) TACR1HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL378394 0.77 TAAR1 (0.51) HPGDNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL379276 0.76 HPGD (0.44) HPGDNPC1RAB9ASMN1; SMN2MEN1
SCHEMBL28231788 0.76 OPRM1 (0.43) TACR1
SCHEMBL378896 0.75 APP (0.50) TACR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed