SCHEMBL3785456

SCHEMBL3785456

NCc1ccc2c(ccn2-c2ccc(F)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.56
LOXL2 Q9Y4K0 1/20 0.46
EPHX2 P34913 1/20 0.41
MGLL Q99685 2/20 0.38
HTR2C P28335 2/20 0.37
HTR2A P28223 1/20 0.37
DRD2 P14416 1/20 0.37
HRH1 P35367 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
ALOX12 P18054 1/20 0.36
RAB9A P51151 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6956593 0.84 KCNH2 (0.56) KCNH2EPHX2MGLLALDH1A1HPGD
SCHEMBL7083302 0.84 KCNH2 (0.56) KCNH2EPHX2MGLLALDH1A1HPGD
SCHEMBL27400803 0.84 PLA2G4A (0.48) KCNH2LOXL2SMN1; SMN2BIRC5TAAR1
SCHEMBL27403901 0.84 TAAR1 (0.44) KCNH2LOXL2HPGDMAOBTAAR1
SCHEMBL6957897 0.81 KCNH2 (0.52) KCNH2EPHX2MGLLALDH1A1HPGD
SCHEMBL5737044 0.80 KCNH2 (0.51) KCNH2EPHX2MGLLALDH1A1HPGD
SCHEMBL4572982 0.79 KCNH2 (0.60) KCNH2EPHX2MGLLHTR2CHTR2A
SCHEMBL30364829 0.79 KCNH2 (0.60) KCNH2EPHX2MGLLHTR2CHTR2A
SCHEMBL5735700 0.77 KCNH2 (0.49) KCNH2EPHX2MGLLALDH1A1HPGD
SCHEMBL27403675 0.77 LOXL2 (0.36) KCNH2LOXL2HTR2CHTR2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010082044-A1 UNSATURATED BICYCLIC HETEROCYCLIC DERIVATIVES AS SMO ANTAGONISTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2010-07-22 WO disclosed