SCHEMBL3787119

SCHEMBL3787119

CCOc1nc(NCc2ccc(F)cc2)nc2nnc(-c3ccc(F)cc3)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 2/20 0.39
MAPT P10636 3/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
EGFR P00533 2/20 0.38
ERBB2 P04626 2/20 0.38
MPO P05164 1/20 0.38
PTGS2 P35354 2/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
GAA P10253 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HTT P42858 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
ATM Q13315 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3782046 0.95 MPO (0.45) KCNH3MAPTMPOPTGS2MEN1
SCHEMBL3776179 0.91 MPO (0.39) MPOMEN1KMT2AHTTCYP1A2
SCHEMBL3780333 0.90 CNR2 (0.48) MAPTEGFRMEN1KMT2AGAA
SCHEMBL3783407 0.89 CA1 (0.42) MAPTCA1CA2CA9PTGS2
SCHEMBL3788039 0.88 MAPT (0.44) KCNH3MAPTPTGS2MEN1KMT2A
SCHEMBL3713217 0.87 KCNH3 (0.41) KCNH3MAPTHTTNPSR1
SCHEMBL3787051 0.84 MEN1 (0.39) KCNH3MAPTMEN1KMT2ACYP1A2
SCHEMBL3785711 0.83 KCNH3 (0.43) KCNH3MAPTMPOMEN1KMT2A
SCHEMBL3782859 0.82 KCNH3 (0.47) KCNH3
SCHEMBL4408548 0.82 MAPT (0.43) KCNH3MAPTCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed