SCHEMBL3783407

SCHEMBL3783407

CCOc1nc(NCc2ccc(S(=O)(=O)NC)cc2)nc2nnc(-c3ccc(F)cc3)nc12

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
CA9 Q16790 4/20 0.42
PTGS2 P35354 9/20 0.41
PTGS1 P23219 1/20 0.39
MAPT P10636 3/20 0.36
RORC P51449 1/20 0.36
GAA P10253 1/20 0.36
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3787119 0.89 KCNH3 (0.39) CA1CA2CA9PTGS2MAPT
SCHEMBL3782046 0.85 MPO (0.45) PTGS2MAPTGAATP53
SCHEMBL3776179 0.81 MPO (0.39)
SCHEMBL3780333 0.80 CNR2 (0.48) MAPTGAATP53
SCHEMBL3781754 0.80 PTGS2 (0.46) PTGS2PTGS1MAPTGAATP53
SCHEMBL3788039 0.79 MAPT (0.44) PTGS2MAPTGAATP53
SCHEMBL3701571 0.79 HRH4 (0.44) PTGS2PTGS1MAPT
SCHEMBL3777960 0.78 GHSR (0.40) PTGS2PTGS1
SCHEMBL3713217 0.78 KCNH3 (0.41) PTGS1MAPT
SCHEMBL4408652 0.76 CA1 (0.53) CA1CA2CA9PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO claimed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed