SCHEMBL3790964

SCHEMBL3790964

Fc1cccc(Cl)c1-c1nc(-c2ccc(Oc3ccccc3)nc2)c[nH]1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGES O14684 10/20 0.43
LTA4H P09960 1/20 0.41
GPR84 Q9NQS5 1/20 0.39
GRM2 Q14416 1/20 0.39
JAK2 O60674 2/20 0.37
ORAI1 Q96D31 2/20 0.37
CTSA P10619 1/20 0.37
BCL2L1 Q07817 1/20 0.37
MCL1 Q07820 1/20 0.37
DGAT1 O75907 1/20 0.36
SOAT1 P35610 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP2C9 P11712 1/20 0.36
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
JAK3 P52333 1/20 0.35
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076592 0.91 ORAI1 (0.41) PTGESORAI1DGAT1
SCHEMBL3795476 0.81 PTGES (0.60) PTGESLTA4HGPR84JAK2ORAI1
SCHEMBL3796320 0.80 PTGES (0.49) PTGESJAK2ORAI1CYP2C9JAK3
SCHEMBL13076230 0.79 PTGES (0.43) PTGESJAK2CYP2C9JAK3
SCHEMBL3802996 0.79 PTGES (0.43) PTGESJAK2
SCHEMBL3795491 0.79 PTGES (0.43) PTGESJAK2
SCHEMBL3796002 0.79 PTGES (0.43) PTGESJAK2ORAI1JAK3
SCHEMBL3796674 0.77 PTGES (0.67) PTGESJAK2CYP2C9
SCHEMBL29662800 0.77 PTGES (0.43) PTGESJAK2CYP2C9JAK3
SCHEMBL13075541 0.77 KDM4E (0.43) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed