SCHEMBL13076592

SCHEMBL13076592

COc1ccc(Oc2ccc(-c3c[nH]c(-c4c(F)cccc4Cl)n3)cn2)cc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ORAI1 Q96D31 2/20 0.41
PTGES O14684 4/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PBRM1 Q86U86 1/20 0.36
MAOB P27338 1/20 0.36
MAPK10 P53779 3/20 0.36
DGAT1 O75907 1/20 0.36
PRKAG1 P54619 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
MAPK8 P45983 1/20 0.35
ALDH1A1 P00352 1/20 0.35
AVPR2 P30518 2/20 0.35
OXTR P30559 2/20 0.35
AVPR1A P37288 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SYK P43405 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3790964 0.91 PTGES (0.43) ORAI1PTGESDGAT1
SCHEMBL3799446 0.82 PTGES (0.52) ORAI1PTGESMAPK10DGAT1
SCHEMBL3796320 0.78 PTGES (0.49) ORAI1PTGES
SCHEMBL13076588 0.77 PBRM1 (0.36) ORAI1PTGESMEN1KMT2APBRM1
SCHEMBL13076230 0.77 PTGES (0.43) PTGES
SCHEMBL3801417 0.76 PTGES (0.48) PTGESDGAT1
SCHEMBL3796002 0.76 PTGES (0.43) ORAI1PTGES
SCHEMBL29662800 0.75 PTGES (0.43) PTGES
SCHEMBL4784907 0.74 RHEB (0.46) PTGESMEN1KMT2AALDH1A1NPC1
SCHEMBL3794879 0.74 PTGES (0.47) ORAI1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed