SCHEMBL3791328

SCHEMBL3791328

COc1cccc(CNC(=O)c2ccc3nn(CC#N)c(=O)n3c2)c1OC

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.52
ROCK1 Q13464 1/20 0.52
POLB P06746 2/20 0.48
NAMPT P43490 1/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
TP53 P04637 1/20 0.44
EPHX2 P34913 1/20 0.42
SCN9A Q15858 1/20 0.42
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
HDAC1 Q13547 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13258566 0.88 ROCK2 (0.54) ROCK2ROCK1POLBNAMPTMAPT
SCHEMBL3794734 0.87 ROCK2 (0.53) ROCK2ROCK1POLBNAMPTMAPT
SCHEMBL3788935 0.82 EPHX2 (0.47) ROCK2ROCK1EPHX2HDAC1
SCHEMBL3793750 0.77 ROCK2 (0.57) ROCK2ROCK1POLBNAMPTMAPT
SCHEMBL3790889 0.71 PPARG (0.52) ROCK2ROCK1EPHX2HPGDHDAC1
SCHEMBL3791605 0.71 EPHX2 (0.49) ROCK2ROCK1EPHX2HDAC1
SCHEMBL3796727 0.70 EPHX2 (0.52) ROCK2ROCK1EPHX2HDAC1
SCHEMBL13258052 0.69 EPHX2 (0.49) ROCK2ROCK1EPHX2HDAC1
SCHEMBL3788362 0.69 EPHX2 (0.49) ROCK2ROCK1EPHX2HDAC1
SCHEMBL3787175 0.69 EPHX2 (0.57) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed