SCHEMBL379145

SCHEMBL379145

c1ccc(CN(Cc2ccccc2)c2ccc(CCCc3ccc(N(Cc4ccccc4)Cc4ccccc4)cc3)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.62
TSHR P16473 2/20 0.53
CNR2 P34972 1/20 0.53
HTR2A P28223 1/20 0.52
NR1H2 P55055 1/20 0.50
NR1H3 Q13133 1/20 0.50
NR3C1 P04150 1/20 0.49
SIGMAR1 Q99720 3/20 0.47
HTR1A P08908 2/20 0.47
ADRA2A P08913 2/20 0.47
ADRA1A P35348 2/20 0.47
OPRM1 P35372 2/20 0.47
DRD3 P35462 2/20 0.47
SLC6A3 Q01959 2/20 0.47
KCNH2 Q12809 2/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4407604 0.91 CYP2C19 (0.67) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL6676662 0.89 CYP2C19 (0.59) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL2960872 0.87 CYP2C19 (0.78) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL3747682 0.84 TDP1 (0.61) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL135570 0.84 CYP2C19 (0.63) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL27886895 0.83 TSHR (0.59) CYP2C19TSHRNR1H2NR1H3SIGMAR1
SCHEMBL10763738 0.83 CYP2C19 (0.67) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL14283665 0.82 CYP2C19 (0.61) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL43183 0.82 TSHR (0.74) CYP2C19TSHRCNR2NR1H2NR1H3
SCHEMBL2011193 0.80 CYP2C19 (0.69) CYP2C19TSHRCNR2NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2666058-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE Ricoh Company Ltd. (JP) 2013-11-27 EP disclosed
EP-2666059-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, AND IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE USING THE ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR Ricoh Company Ltd. (JP) 2013-11-27 EP disclosed
EP-2616883-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE Ricoh Company Ltd. (JP) 2013-07-24 EP disclosed
WO-2012099181-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE RICOH COMPANY, LTD. (JP) 2012-07-26 WO disclosed
WO-2012099182-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, AND IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE USING THE ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR RICOH COMPANY, LTD. (JP) 2012-07-26 WO disclosed
WO-2012036295-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, IMAGE FORMING METHOD, IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE RICOH COMPANY, LTD. (JP) 2012-03-22 WO disclosed
EP-2409196-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, PRODUCTION METHOD OF THE SAME,IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE Ricoh Company, Ltd. (JP) 2012-01-25 EP disclosed
WO-2010107130-A1 ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR, PRODUCTION METHOD OF THE SAME,IMAGE FORMING APPARATUS, AND PROCESS CARTRIDGE RICOH COMPANY, LTD. (JP) 2010-09-23 WO disclosed